Kiwon lafiyaShirye-shirye

"Moxifloxacin": umarnin don amfani, description, abun da ke ciki

A medicament "Moxifloxacin" pharmacological sakamako na wanda za a tattauna nan, tana nufin rukuni na quinolones. A kayan aiki yana da wani bactericidal, antibacterial sakamako. Next, mun tattauna abin da ya ƙunshi wani magani "Moxifloxacin". Umarnin don amfani, analogues ma za a nuna a cikin labarin.

sakamako

Yadda yake aiki wakili "Moxifloxacin"? Description da miyagun ƙwayoyi kamata a fara da bayanin irin inji na tasirinta a kan kwayoyin cuta. Bactericidal sakamako na nufin hade tare da hanawa (danniya) na kwayan topoisomerase IV kuma II. Wannan, bi da bi, take kaiwa zuwa disturbances a cikin kwafi matakai na kwafi, DNA gyara biosynthesis da ake dasu Kwayoyin. A sakamakon haka, akwai zo ga halaka su. Medicament "Moxifloxacin" umurci manual bayyana a matsayin m bakan kwayoyin.

juriya

A kan antibacterial aiki da kwayoyi "Moxifloxacin" ba zai shafi sunadaran da cewa tsokana da juriya ga tetracyclines, macrolides, aminoglycosides, cephalosporins da penicillins. Yana ba da alama sosai da kuma sakamako na giciye-juriya. Har yanzu, lokuta da jini da kwanciyar hankali da aka ba gano. Drug juriya "Moxifloxacin" tasowa quite sannu a hankali da mahara maye gurbi.

kewayon aiki

Na nufin "Moxifloxacin (umurci manual - hujja) rinjayar da yawa damuwa na gram-tabbatacce kuma gram-korau kwayoyin cuta, acid-sauri kwayoyin cuta, anaerobes, atypical kwayoyin (wato Mycoplasma, chlamydia, da dai sauransu), da kuma kwayoyin da suke resistant zuwa macrolide da beta-lactam kwayoyin kwayoyi .

tsotsa

Lokacin da samun da na baka sha na da miyagun ƙwayoyi "Moxifloxacin" m, kuma kusan ya cika. Cikakkar bioavailability lokacin gudanar intravenously da ake ji a cikin gida - da oda na 91%. Lokacin gudanar da baki (50-1200 MG kashi, 600 MG / rana for 10 days) mikakke pharmacokinetics da miyagun ƙwayoyi. Matsakaicin taro da 400 MG lura bayan 0.5-4 hours. A lokacin da shafi lokaci guda tare da abinci cimma wata karuwa a cikin tsawon lokaci Cmax (sa'o'i biyu), kuma ta rage ta game da 16%. Duration sha haka ya zauna canzawa. Duk da haka, wadannan bayanan da ba su da na asibiti darajar da damar yin amfani da miyagun ƙwayoyi "Moxifloxacin", ko da kuwa da abinci. Wadannan guda igiyar jini jiko na 400 MG ga sa'a iyakar taro ya auku a karshen jiko.

rarraba

A cikin kwanaki uku na aikace-aikace da aka kai ma'auni. Dauri ga jini sunadaran - game da 45%. Yana Notes fairly m rarraba da miyagun ƙwayoyi "Moxifloxacin" gabobin da kyallen takarda. Highest yawa ne a cikin huhu da nama da kuma bronchi mucous, fata da kuma subcutaneous Tsarin, sinuses, kumburi foci. A yau da kuma interstitial ruwa medicament da aka samu a Sakakken sunadarai, free form. Its maida hankali ne ya fi a jini. Tare da wannan magani da aka samu a yawa a gabobin peritoneum kyallen takarda kaciyar mata gabobin da kuma a cikin peritoneal ruwa.

metabolism

Medicine "Moxifloxacin" (bayanin da miyagun ƙwayoyi a annotation data qunshi bayanai) ya wuce na biyu biotransformation lokaci. Koda tukar tumbi aiwatar da tsarin da hanji mai sãkẽwa ba a cikin nau'i na sulpho mahadi da kuma m glucuronide. A metabolites da ake samu a jini. Su maida hankali ƙananan fiye da na asali fili. Nazarin ya nuna cewa wadannan ƙasƙanci kayayyakin ba su da wani korau tasiri a jiki.

Na nufin "Moxifloxacin", daga abin da aka wajabta?

Da miyagun ƙwayoyi bada shawarar ga cututtuka mai kumburi pathologies a manya tsokane ta kwayoyin ciwon ji na ƙwarai, a nan. A musamman, da karatu da lãbãri a wani exacerbation na kullum mashako kwarara, m sinusitis, al'umma-samu ciwon huhu (lalacewa ta hanyar damuwa da kwayoyin cuta exhibiting mahara juriya a t. H. The kwayoyin). Na nufin "Moxifloxacin" umarnin don amfani da shawarar ga cututtuka na m nama da kuma fata, subcutaneous Tsarin wuya raunuka (kamu da ciwon sukari kafar kazalika), da kuma ciki-ciki cututtuka (polymorphic matakai, intraperitoneal abscesses da sauransu). Da ake sa lokacin da medicament daga Streptococcus pneumoniae resistant ga mahara antibacterials, ciki har da gaban resistant damuwa penicillin, biyu ko fiye kungiyoyin na kwayoyi na biyu ƙarni cephalosporins, macrolides, tetracyclines. By alamomi kuma sun hada da kumburi raunuka a pelvic gabobin uncomplicated yanayi. Lokacin da endometritis da salpingitis an kuma karfafa la'akari da nufin (kamar yadda aka nuna ta a haɗe zuwa da miyagun ƙwayoyi "Moxifloxacin" umarnin don amfani). Ido saukad wajabta kwayan conjunctivitis, tsokane ta microorganisms kula da medicament. Haka ma wajibi ne don la'akari da data kasance magani daga cututtuka pathologies shugabanci.

Medicament "Moxifloxacin": da sashi da kuma hanya da gwamnati

Kudi kaddamarda a cikin gida (baki) da kuma intravenously. . Duration na lura da medicament "Moxifloxacin", sashi na wanda - 400 MG / rana, dangane da irin cuta da kuma ta mai tsanani, kazalika da lura warkewa sakamako:

  • Exacerbation na kullum mashako shakka - 5-10 kwana.
  • Community-samu ciwon huhu - 7-14 kwanaki bi da bi far (igiyar jini biyo ta baka ci).
  • Haduwar jijiyoci mai taushi, fata (uncomplicated), kuma m sinusitis - 7 kwanaki.
  • Lokacin da ciki-ciki cututtuka (rikitarwa) - 5-14 kwanaki bi da bi far.
  • Lokacin da wuya raunuka da kuma subcutaneous Tsarin fata - 7-21 kwana.
  • A kumburi pathologies na pelvic gabobin - 14 days.

Don ƙarin bayani, ta kunshi a haɗe zuwa da miyagun ƙwayoyi "Moxifloxacin" umurci manual. Allunan kamata ba a yarda ya tauna. Wanke saukar da ruwa wajibi ne a wani karamin girma.

gida amfani

Medicine "Moxifloxacin" (saukad da) za a iya gudanar da su marasa lafiya da shekara. Yi ya nuna cewa kyautata zo a kan rana ta biyar. Bayan da ya kamata ka ci gaba da jiyya ga wata kwanaki 2-3. Marasa lafiya a cikin shafa ido shuka a drop sau uku a rana. Idan akwai wani sakamako na kwanaki biyar kamata tada tambaya da daidaitar far ko ganewar asali. A tsawon lokaci da magani dogara a kan bacteriological da kuma na asibiti hanya da kuma tsanani daga cikin Pathology.

Bugu da ari a kan for jiko bayani

Medicament "Moxifloxacin" umurci manual bada shawarar cewa ka shigar da awa daya. Da miyagun ƙwayoyi haka zai iya zama a cikin undiluted ko a diluted form. A bayani da jituwa tare da sodium chloride 0.9%, ruwa ga allura, dextrose bayani a maida hankali 10% kuma 40%, 20% xylitol, "Ringer". Yi amfani kawai share taya. Bayan dilution na medicament zauna barga for kwana a dakin da zazzabi. Bai kamata a kiyaye a cikin firiji wajen. Idan jiko da ake gudanar da sauran jamiái, kowanne daga wanda aka gudanar dabam.

illa

Saboda lura magani "Moxifloxacin" kusantar wajen samar da fungal cututtuka, leukopenia, anemia, thrombocytopenia. A wasu lokuta, da far akwai wani karuwa a prothrombin lokaci, thromboplastin yawa canza. A wasu marasa lafiya da miyagun ƙwayoyi zai iya sa rashin lafiyan halayen, laryngeal edema, urticaria, anaphylactic buga, pruritus, eosinophilia, kurji. A rare lokuta, akwai hyperglycemia, hyperlipidemia, hyperuricemia. A lura da m shafi tunanin mutum da cuta. A musamman, marasa lafiya na iya fuskanci Hyperactivity, tashin hankali, ciki, depersonalization, hallucinations, psychotic halayen, tare da suicidal tunani. Common illa hada da ciwon kai, dizziness, tremors, drowsiness, da ruɗewa, dandano ƙwarai cuta, barci disturbances, disorientation. A wasu lokuta, a lokacin jiyya da magani iya sosai daidaituwa, seizures, tare da daban-daban na asibiti manifestations, hypoesthesia, cuta na ji na wari. A yawan marasa lafiya da worsening da magana, da hankali, na gefe neuropathy, ɓacin hankali, polyneuropathy. A lokacin da shafi topically, hangen nesa da iya deteriorate har ta hasãra. Duk da haka, da karshen an dauke su a dõgẽwa yanayin.

Tasiri a zuciya da jijiyoyin jini tsarin

Sashe na da tasiri da aikace-aikace da miyagun ƙwayoyi "Moxifloxacin" ne QT-tazara da tsawaita a cikin marasa lafiya da hypokalemia, palpitations, vasodilation, tachycardia. Rare illa hada da hauhawar jini da kuma hypotension, na ramin zuciya tachyarrhythmias, syncope. Sosai da wuya ya lura sakamakon bugun zuciya. Šauki kagaggun hankula ga mutane predisposed zuwa m ischemia, bradycardia (asibiti gagarumin).

Tasiri a kan sauran tsarin da kuma gabobin

A wasu lokuta, da miyagun ƙwayoyi iya haifar da nakasa daga 'ya'yan numfashi, ciki har da asthmatic yanayin. A yawan marasa lafiya aka lura cuta a cikin narkewa kamar fili. A musamman, kan bango na lura-ullowar tashin zuciya, amai, zawo, ciki zafi. In mun gwada 'yan illa suna dauke matalauta ci, dyspepsia, flatulence, gastroenteritis (sai dai erosive), maƙarƙashiya. Wasu marasa lafiya da aka gano stomatitis, dysphagia, pseudomembranous colitis. A far zai yiwuwa kara a transaminases, hanta tabarbarewa, ci gaban fulminant hepatitis, hanta gazawar manyan zuwa rai barazana. Sosai da wuya ya lura bullous cutaneous halayen (mai guba epidermal necrolysis, Stevens-Johnson ciwo). Wasu marasa lafiya samu myalgia, arthralgia, convulsions, ta ƙara tsoka sautin, tendonitis, tsoka rauni. agara ruptures iya faruwa a rare lokuta, amosanin gabbai, Gait tashin hankali a sakamakon lalacewar da musculoskeletal tsarin. Marasa lafiya a kan magani da magani iya zama ya lura da cuta daga cikin urinary tsarin. A musamman, alama dehydration (tsokani zawo ko karu a ruwa girma cinye), koda tabarbarewa, insufficiency. Common illa hada sweating, nonspecific zafi, malaise. A cikin igiyar jini m thrombophlebitis ko phlebitis.

Wanda ba a sanya wa hanyar?

A magani "Moxifloxacin" contraindications ne kamar haka:

  • Agara Pathology a tarihi cewa ci gaba a sakamakon far quinolone maganin rigakafi kungiyar.
  • Availability elongate QT-tazara (nakasar ko samu).
  • Electrolyte disturbances (musamman hypokalemia uncorrected).
  • Bradycardia (asibiti gagarumin).
  • Zuciya rashin cin nasara tare da rage ejection aiki a hagu ventricle.
  • Keta zuciya kari (a tarihi).

Lokacin da lactose rashin ha} uri, glucose-galactose malabsorption, lactase rashi ne kuma ba da shawarar medicament "Moxifloxacin" (miyagun ƙwayoyi abun da ke ciki qunshi lactose, saboda haka pathologies da aka ambata ana kunshe a cikin jerin). Ba sanya nufin ciki ko lactating. Allunan, kuma da bayani da aka yarda to manufa marasa lafiya shekaru 18 da haihuwa. Shawarar da miyagun ƙwayoyi a hali na hypersensitivity da aka gyara.

lokuta na musamman

Tsanaki ake bukata a cikin saduwa da miyagun ƙwayoyi ga marasa lafiya da tsakiya m tsarin munanan cewa predispose ga ci gaban seizures. A hadarin kungiyar hada da marasa lafiya da proarrhythmic jihohi. Wadannan sun hada da, musamman, sun hada da m ischemia, musamman a cikin tsofaffi da kuma mata. Har ila yau tsayar da taka tsantsan a marasa lafiya tare da hanta cirrhosis. sashi gyara iya da ake bukata a lokacin lokaci guda far nufin ragewan da taro na potassium.

Don ƙarin bayani,

Yi ya nuna cewa da miyagun ƙwayoyi ne da jure a da yawa marasa lafiya. Kwararru sau da yawa rubũta da kayan aiki ga cututtuka raunuka. Wannan shi ne saboda cewa da miyagun ƙwayoyi yana da wani gwada da high dace da yawa kwayoyin. Duk da haka, akwai ko da yaushe hadarin illa, wanda ake hada da samfurin yayi kashedin "Moxifloxacin" umurci manual. Analogs da miyagun ƙwayoyi a hali na bukatar kamata karba likita akayi daban-daban. Sauya kayan aiki iya irin wannan kwayoyi a matsayin: "Avelox", "Vigamoks", "Rotomoks", "Moksifur", "Moksin" da sauransu. Lokacin da illar, mai kaifi tabarbarewar da kuma abin da ya faru na cututtuka da cewa ba su bayyana a cikin summary, dole ne ka nemi likita nan da nan hankali. Lokacin amfani da saukad da ya kamata kauce lamba tare da matsanancin yawa daga cikin miyagun ƙwayoyi ta idanu. Idan wannan ya faru, za ka bukatar da sauri tare da yalwa da ruwa. A hali na yawan abin sama kayan haɓɓaka aiki na gefe effects.

a ƙarshe

Da miyagun ƙwayoyi "Moxifloxacin" dauke isasshe m antibacterial. A dangane da wannan musamman shi ba da shawarar karya da ganin likita. A musamman, shi ya shafi yawan da kuma mita na aikace-aikace wajen. Kada ku ƙẽtare sashi. Igiyar jini allura kamata a da za'ayi a cikin wani musamman nazari ta ƙwararren ma'aikacin wanda za su iya taimaka idan ya cancanta. Ya kamata ka ba kai-medicate. A rashin sakamakon far wajibi ne don ganin likita. Kamar kafin amfani da miyagun ƙwayoyi "Moxifloxacin" ya kamata a hankali karanta umarnin.

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