Kiwon lafiya, Shirye-shirye
"Mirapex": umarnin don amfani, description, reviews
A wannan labarin, za ka koyi dukan game da shirye-shiryen "mirapex": da yadda za a maye gurbin wannan miyagun ƙwayoyi, abin da yake tasirinta, contraindications, illa, musamman umarnin da hannunsa. Wadannan kwayoyi zai iya sa mahaukaci hali da kuma tasiri a kan haƙuri ta mayar da martani. Saboda haka, kafin shan wannan magani "mirapex" umarnin don amfani da ya kamata a hankali karatu. Mun kuma gaya maka game da karfinsu na wadannan kwayoyi da sauran kwayoyi.
Tsawo "mirapex": janar bayani game da miyagun ƙwayoyi da kuma alamomi ga yin amfani da
The aiki abu na cikin shirye-shiryen "mirapex" ne pramipexole. Karin aka gyara Allunan: povidone, mannitol, sitaci, aerosil, magnesium stearate.
Tare da wannan magani far da aka kwashe idiopathic (mai zaman kanta da sauran raunuka) ciwo na "m kafafu" da kuma Parkinson ya cutar, kazalika da sauran mai ladabi mota da kuma extrapyramidal cuta.
Product: kwayoyi "mirapex PD" 3 MG, 4.5 MG, 1.5 MG, 0.75 MG, 0,375 MG. Suna cushe a blisters na 10 guda, sa'an nan a cikin kwali kwalaye.
fari kwayoyi. Bã su da wani beveled baki da lebur siffar a garesu, daya daga wanda yana da wani babban hadarin.
Allunan ya kamata a dauka baki, ko da kuwa abinci. Ci miyagun ƙwayoyi ne a yarda a kowane lokaci. A wannan yanayin, shi ya kamata a wanke saukar da ruwa. Nagari kullum kashi ne zuwa kashi uku, saukarwa.
Ginshikai na mataki (pharmacodynamics) "mirapex" Allunan
Tasiri pramipexole abu wanda qunshi shiri "mirapex" musamman da tare da babban selectivity kara habaka da martani na subgroup na dopamine rabe D2. Godiya ga shi, cika wa cikin rashin jiki aiki a yanayin saukan Parkinson ta cutar. Wannan shi ne saboda kunnawa da dopamine rabe a striatum. Kamar wancan pramipexole hana degeneration na neurons cewa ya auku saboda neurotoxicity ko ischemia. Yana damuarn ko rage kudi na kira, metabolism, da kuma sakin dopamine. Godiya ga pramipexole neurons an kare daga mai guba effects na anti-Parkinson jamiái "Levodopa". Har ila yau, saboda tasirinta rage-rage prolactin (kashi-dogara).
A cikin hali na shafe tsawon amfani da kwayoyi "mirapex" domin lura da Parkinson ya cutar (fiye da shekaru uku) da kuma ciwo na "m kafafu" (fiye da shekara) bai saukar da rage yadda ya dace da pramipexole.
Biochemical matakai shafe shiri "mirapex 'a haƙuri ta jiki (pharmacokinetics)
Active abu "mirapex" da miyagun ƙwayoyi ne gaba daya da kuma hanzari tunawa bayan baka gwamnati. Iyãwarsa ga assimilation (bioavailability) ne kusan cikakkar - fiye da 90%. Matsakaicin taro na miyagun ƙwayoyi a jini lura bayan 1-3 hours bayan cin abinci. A abinci pramipexole Absorption Rate rage-rage. A wannan yanayin, da adadin digestible abinci ba ya canja.
C sunadaran ta ɗaure pramipexole dan kadan (kasa da 20%). Yana yana da babban rarraba girma - 400 lita, wanda ke nufin cewa maida hankali a cikin jini ne low. Don a kananan har fallasa da miyagun ƙwayoyi metabolism tsari. Aƙalla 90% na kashi "mirapex" katsin excreted da kodan, tare da 80% - canzawa. Tumbi pramipexole da aka samu a wani adadin na kasa da 2% na cinye adadin da miyagun ƙwayoyi. Nama da kuma jiki ruwaye aka tsarkake daga "mirapex" Allunan a wani talakawan kudi na 500 ml / min.
Amfani "mirapex" miyagun ƙwayoyi a lokacin daukar ciki
Zan iya amfani da lokacin daukar ciki "mirapex" kwamfutar hannu? Umurnai na yin amfani da miyagun ƙwayoyi da shi a fili cewa da tasiri na da miyagun ƙwayoyi a kan ci gaban da tayin a cikin mahaifar, lactation ba a bincika.
Tukar tumbi da pramipexole cikin ƙirjinka madara ba a karatu. Daya iya kawai zaton cewa abu zai iya hana lactation, tun inhibits samar luteotrophic hormone. Saboda haka, kada ku riƙi "mirapex" kwaya a lokacin shayarwa.
A lokacin daukar ciki, da miyagun ƙwayoyi ya kamata a dauka kawai idan m amfani zuwa ga uwar marasa nan gaba hadarin da tayin.
Contraindications ga yin amfani da Allunan 'mirapex "
Drug "mirapex" ba za a iya dauka a cikin hali na hypersensitivity zuwa pramipexole, kazalika da mutane suka yi ba ta kai shekaru 18 da haihuwa.
Tare da musamman hankali bada shawarar yin amfani da Allunan, a karkashin rage hawan jini da kuma koda gazawar.
Side effects "mirapex" miyagun ƙwayoyi a kan m tsarin
Shiri "mirapex" - Allunan wanda zai iya sa da juyayi tsarin wadannan halayen:
- rikice.
- wuce kima craving for barci ko rashin kyawunsu;
- hallucinations.
- ɓacin hankali.
- asthenia.
- dizziness.
- extrapyramidal ciwo.
- hypoesthesia.
- tsãwa;
- myoclonus.
- dystonia.
- ciki;
- delirium.
- suicidal nufi.
- hypokinesia.
- ataxia.
- tashin hankali.
- neuroleptic m ciwo.
Last gani a cikin nau'i na hyperthermia, disturbances na sani da tunani, tsoka rigidity, autonomic lability, akathisia.
Side effects na kwayoyi "mirapex" a kan sauran tsarin na jikin mutum
Musculoskeletal tsarin iya amsa ga yin amfani da magunguna "mirapex" wannan manifestations:
- hypertonic tsokoki, da convulsions, twitching.
- abin da ya faru na amosanin gabbai, myasthenia gravis ko bursitis.
- zafi a cikin kirji, wuyansa, ko kashin baya (a cikin lumbosacral).
Su kuma iya faruwa saɓani a cikin narkewa kamar tsarin. Lokacin da wannan ya auku:
- asarar ci.
- maƙarƙashiya.
- tashin zuciya.
- dyspepsia.
- flatulence.
- zawo.
- amai.
- bushe baki.
- yankan ji a ciki.
Numfashi liyafar "mirapex" da miyagun ƙwayoyi iya haifar da ci gaban sinusitis, pharyngitis, rhinitis, mura-kamar ciwo. Shi ne kuma zai yiwu ya faru na shortness na numfashi, ta ƙara tari da kuma murya canji.
Mene ne sakamako a kan zuciya da jijiyoyin jini tsarin "mirapex" kwamfutar hannu? Umurnai na yin amfani da miyagun ƙwayoyi sanar da game da yiwu ci gaba tachycardia, arrhythmia, angina pectoris, orthostatic hypotension.
Sauran illa
Lokacin da samun da miyagun ƙwayoyi "mirapex" irin matsalolin da za su iya faruwa a cikin urogenital tsarin, kamar yadda mafi m hanji ƙungiyoyi, kamuwa da cuta. Kamar haka ko da ya kamata asarar libido da kuma iko.
Bugu da kari, kana iya samun biyu hangen nesa, cataract, conjunctivitis, inna da masauki, allergies, kuma illa ji, da intraocular matsa lamba.
Sauran m halayen na jiki:
- retroperitoneal fibrosis.
- pleural effusion.
- na huhu infiltration.
- nauyi asara.
- gefe edema.
Sashi da Administration "mirapex" Allunan
Don amfani da miyagun ƙwayoyi da kuke bukata a ciki, kullum sau 3. Harufan kashi "mirapex PD" Allunan - 0,375 MG da rana. A hankali kara yawan miyagun ƙwayoyi zama dole (kowane 7 days) to samu da ake so warkewa sakamako. A mako na biyu na magani kowace rana kamata a ƙone su da 0.75 MG a cikin na uku - a 1,5 MG a karo na hudu - ta 2.25 MG a cikin na biyar bukatar sha magani "mirapex" 3 MG da kullum, a kan shida - 3,75 MG, na bakwai - 4.5 MG.
A kullum na koda gazawar, da sashi ne gyara dangane da wasan kwaikwayon matakin na creatinine yarda. A daidai adadin da miyagun ƙwayoyi ya kamata a nada wani likita.
Sakamakon yawan abin sama kwaya "mirapex"
Idan ka yi amfani da "mirapex" miyagun ƙwayoyi sashi aka karya, wadannan cututtuka zai iya faruwa yiwuwa hallucinations, hyperkinesia, tashin zuciya da amai, rage hawan jini da kuma arousal.
Domin wannan halin da ake ciki, da maganin guba da aka ba shigar. Lokuta da miyagun ƙwayoyi yawan abin sama "mirapex" ba gyarawa. Nagari symptomatic far, ciki lavage kuma tsauri kallo. Idan akwai alamun wani yawan abin sama da zumudi na tsakiya m tsarin, ya zama dole su yi amfani da shirye-shirye, neuroleptics.
Interactions Allunan "mirapex" tare da wasu kwayoyi
Pramipexole hade jini gina jiki dan kadan da kuma biotransformation. Saboda haka, ta hulda da sauran kwayoyi da shafi wadannan matakai ne da kamar wuya.
Kwayoyi da hana ko kashe samar da aiki abubuwa ko cationic samovyvodyaschiesya ta hanyar da na koda tubules, za a iya amsa tare da kwayoyi "mirapex". Umurnai na amfani bayyana cewa, a wannan yanayin da gudun rage bayyananne tsarkakewa tsokoki da nazarin halittu ruwaye ko daga duka medicaments ko daya daga cikinsu.
Idan lokaci guda tare da kwayoyi 'mirapex "amfani da wadannan kwayoyi, ya kamata ka kula da yiwu hallucinations, dyskinesia, agitation. Idan wadannan alamu faruwa, da sashi daga cikin miyagun ƙwayoyi ya kamata a rage.
Karfinsu Allunan "mirapex" tare da kwayoyi "Amantadine" da "L-dopa"
Menene ya faru sa'ad da hada liyafar "Levodopa" kwayoyi da kuma "selegiline" kwayoyi "mirapex PD"? Umarni ya furta cewa, pharmacokinetics na aiki wakili ba zai tasiri ba na farko kuma na biyu. A lokaci guda a kan cikakken assimilation da tukar tumbi da miyagun ƙwayoyi a wani halitta hanya "Levodopa" kwamfutar hannu "mirapex" an ba a gane.
Pramipexole aka ba karatu da hulda da miyagun ƙwayoyi "Amantadine". Amma karfinsu ne zai yiwu a far, tun suna da kama da sunadaran da tukar tumbi.
Lokacin da kashi "mirapex" shiri ya karu, da aikace-aikace adadin "Levodopa" da shawarar a rage. Yawan sauran antiparkinsonian kwayoyi dole ne a kiyaye kullum a wannan matakin.
Features Karfinsu shiri "mirapex" tare da wasu kwayoyi
Saboda da yiwuwar tarawa effects tare da matsananci hankali bada shawarar yin amfani da Allunan "mirapex" a hade tare da sedatives, barasa, da kuma kwayoyi da cewa taimaka wajen kara pramipexole maida hankali a cikin jini (msl, wani magani "Cimetidine").
Specific shiriya a cikin yin amfani da "mirapex" Allunan
Muna kwatanta da miyagun ƙwayoyi ba da shawarar a yi a tare da antipsychotics.
A lura da dopamine agonist sani illa su rikice da kuma hallucinations. A lokuta da "mirapex" Allunan a hade tare da miyagun ƙwayoyi "Levodopa" irin munanan kasance mafi m, a cikin hãlãye daga baya da cutar fiye da a farkon monotherapy.
A likita dole ne a sanar da haƙuri da zai yiwu ya faru na gani hallucinations. Wannan gefen sakamako rinjayar da ikon fitar da motoci da yin alhakin yanke shawara.
A kaifi an daina Allunan a cikin hali na Parkinson ya cutar da aka gano bayyanar cututtuka da yayi kama neuroleptic m ciwo.
Anomalous hali a cikin yin amfani da "mirapex" miyagun ƙwayoyi
Marasa lafiya da waɗanda kula da su, shi ne wajibi ne su san cewa liyafar na dopaminergic kwayoyi, ciki har da "mirapex" Allunan (reviews tabbatar da wannan), sau da yawa yana sa mahaukaci hali na haƙuri. Za ka iya samun hyperphagia (overeating buri), pathological shopping (m so in yi yawa sayayya), na kullum cãca, kuma hypersexuality. A irin haka shi wajibi ne don rage sashi daga cikin miyagun ƙwayoyi ko hankali daina shan shi.
Tsanaki a cikin yin amfani da "mirapex" Allunan
Medicine "mirapex" Ya kamata a cinye tare da taka tsantsan ga marasa lafiya da gaban tsanani cututtuka na zuciya da jijiyoyin jini tsarin. A gudanar da far da dopaminergic kwayoyi akwai wani hadarin orthostatic hypotension. Saboda haka, a jini iko, musamman a farko mataki na magani.
Lokacin da na gani hanawa ne dole a kai a kai duba shi nan da nan bayan da nada Allunan "mirapex" da kuma kara tsare jinkiri.
Marasa lafiya ya kamata a ba da gaskiya cewa miyagun ƙwayoyi iya samun magani mai kantad da hankali sakamako. Akwai sun kasance lokuta na kwatsam barci da kuma wuce kima sleepiness a lokacin da rana ayyukan. Ciki har da wannan na iya faruwa a kowane lokaci a gudanar da hadadden kayan aiki, ko tuki motocin.
The yiwuwar tasowa melanoma
A sakamakon ANNOBA karatu sun nuna cewa marasa lafiya da Parkinson ya cutar ne a hadarin melanoma. Shin shi cikin hanyar da wannan cuta, ko wasu dalilai, kamar yin amfani da "mirapex" da miyagun ƙwayoyi ba a kafa.
Ƙarfafa na ciwo na "m kafafu"
Ta yaya ciwo na "m kafafu" miyagun ƙwayoyi "mirapex"? Shedu nuna cewa dopaminergic kwayoyi iya inganta shi. Wannan yana bayyana a cikin nau'i na baya farko na bayyanar cututtuka da yamma ciwo da kuma wani lokacin da rana. A wannan yanayin, da cututtuka yada zuwa wasu gabar jiki. The gudanar for 26 makonni a asibiti sarrafawa binciken, wanda aka tsara don nazarin wannan sakamako, wani gagarumin bambanci tsakanin pramipexole da placebo kungiyoyin a inganta fasali na ciwo da aka gano.
Storage yanayi da kuma shiryayye rai
"Mirapex" kwamfutar hannu tana nufin wani shiri na jerin B. Store suka kasance a cikin wani duhu wuri. A wannan yanayin da dakin da zazzabi kada wuce 30 ° C.
Shiryayye-rai da miyagun ƙwayoyi - watanni 36 (3 years) daga kwanan watan da samar.
Da amfani da "mirapex" Allunan a cikin shimfiɗar jariri, da yanayi na saya
Da miyagun ƙwayoyi ne contraindicated don amfani a yara. Izni da aka kãwo wa mutane samun Allunan, wanda sun kai shekaru 18 da haihuwa. Medicine "mirapex" saki a Pharmacy a gabatar da takardar sayen magani.
Drug analogues "mirapex"
Ba za ka iya, domin duk abin da dalili, don saya da kwamfutar hannu ne "mirapex"? Abin da zai iya maye gurbin da miyagun ƙwayoyi, ya kamata ka gaya wa harhaɗa magunguna ko likita. Kuma muna bayar da wadannan analogues.
- "Motopram" kwayoyi. Alamomi ga yin amfani: Parkinson ta cutar. Yana za a iya yi shi kadai, ko a hade da magani magani 'levodopa'. Yana kuma amfani da tsanani ko matsakaici idiopathic nau'i na ciwo na "m kafafu".
- "Oprimeya" kwayoyi. Manufa: antiparkinsonian magani stimulant dopaminergic watsa a tsakiya m tsarin.
- "Pramipexole" kwayoyi. A warkewa wakili a yi amfani da Parkinson ta cutar. An yi imani da cewa ginshikai na mataki ne kai tsaye da nasaba da ikon da wani abu pramipexole ta da dopamine rabe a striatum.
Allunan "mirapex" - analogues ko asali? Babu kai!
A cikin sama da aka jera kayayyakin, wanda suke analogues na 'mirapex "Allunan. Suna da wannan musamman, kasa da kasa wadanda ba na mallakar tajirai sunan (ko ATC-code), wanda aka shawarar da WHO (World Health Organization).
Idan kana bukatar ka sha magani ta yin amfani da Allunan "mirapex" analogs kuma iya zama mai girma madadin. Amma kafin ka maye gurbin nada wajen far, tabbata tuntubar da gwani. Babu wani hali da ba kai! Wannan zai iya haifar da komowar mummunan sakamakon for your kiwon lafiya.
Gargadi! Wannan labarin ne mai bayanin "mirapex" shiri ne suna goyon bayan da kuma Sauki version na aikin hukuma umarnin don amfani. Drug bayanai da aka gabatar ga manufar review. A wani hali ba yin amfani da shi a matsayin mai shiryarwa zuwa kai-magani.
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