Kiwon lafiya, Shirye-shirye
Da miyagun ƙwayoyi "Pentas": umarnin don amfani, analogs da kuma sake dubawa
A wani kashi na wajabta magani "Pentas"? Umurnai na amfani, da kuma sake dubawa na miyagun ƙwayoyi da aka bayyana a kasa. Har ila yau a cikin kayan labarin bayar da bayanai game da siffofin saki na miyagun ƙwayoyi da kuma da kaddarorin.
A abun da ke ciki, siffar medicament
Akwai da dama siffofin saki dauke magunguna. Mun gabatar da su a yanzu.
Shiri "pentasil" - Allunan (500 MG, 100 MG) shafe tsawon mataki. Su farar da wani grayish tinge, kazalika da yawa faci na haske launin ruwan kasa, da daidai zagaye siffar, tare da Valium, bevel da inscriptions a garesu.
The aiki kashi na wannan magani ne mesalazine. Har ila yau da nufin ne a cikin nau'i na m sinadaran povidone, ethylcellulose, magnesium stearate, talc, da kuma microcrystalline cellulose.
A sayar da miyagun ƙwayoyi "Pentas" (Allunan), wani photo na wanda aka gabatar a cikin labarin da aka kawota a bororo fakitoci da suke a cikin takarda cartons.
Ya kamata kuma a lura da cewa, batun medicament za a iya saya a cikin nau'i na suppositories, ci-saki granules da rectal dakatar.
Pharmacology magani
Mene ne magani ga "Pentas"? Umurnai na amfani furta cewa, wannan wakili da anti-mai kumburi mataki da kuma amfani da su bi ulcerative colitis da Crohn ta cuta.
Anti-mai kumburi Properties daga cikin miyagun ƙwayoyi bayyana ne kawai ga gida amfani. Wannan mataki ne ya sa ta kira na leukotrienes da prostaglandins, kazalika da hanawa na lipoxygenase aiki (neutrophil). Bugu da ƙari kuma, da kayan aiki ne iya retard mugunya immunoglobulin da lymphocytes da kuma hana degranulation, kuma phagocytosis na neutrophil hijirarsa.
Musamman gastrointestinal jamiái
A medicament "pentasil" (kwamfutar hannu), da abun da ke ciki na wanda aka gabatar a sama, farfado furta antibacterial aiki da wasu cocci da Escherichia coli. Har ila yau, yana da wani antioxidant sakamako saboda da ikon kisa da aiki abu da free radicals (oxygen) da kuma hallakar da su.
Dace na amfani da wannan kayan aiki ƙwarai rage hadarin koma dawowan cutar a Crohn ta cuta, ciki har da mutane da ileitis (tare da wani dogon cuta duration).
Ka'idar aiki na likitanci da wuraren
Ta yaya miyagun ƙwayoyi "Pentas"? Umarnin a kan aikace-aikace shelanta cewa warkewa sakamako daga cikin miyagun ƙwayoyi ne nan da nan bayan Topical mesalazine lamba tare da hanji mucosa.
Bayan shan baka hannu yana nufin nan da nan disintegrates a microgranules wanda aiki a matsayin raba siffofin da ci aiki abu saki - mesalazine. Wannan na samar da wani kyau miyagun ƙwayoyi domin tsakanin 12- zuwa dubura a duk PH dabi'u.
Pharmacokinetics nufin
Ta yaya sha na da miyagun ƙwayoyi "Pentas"? Umurnai na yin amfani da rahotannin da ke cewa microgranules na rududdugaggun Allunan 12 ya kai duodenum a cikin ta farko 60 minutes.
Aƙalla 30-50% na wani tunawa sashi daga cikin miyagun ƙwayoyi a cikin kananan hanji. Communication mesalazine da jini da sunadarai ne 43% da kuma acid N-acetyl-biyar-aminosalicylic - 73-85%.
Mesalazine Irinta ba shiga cikin BBB. Tarawa miyagun ƙwayoyi Properties suna bayyana ne kawai a lokacin da yin amfani da high allurai (game da 1500 MG da rana).
Acetylation mesalazine aka fallasa a cikin hanji mucosa da kuma hanta. Wannan abu da aka samu daga fitsari, nono da madara da kuma tumbi.
Alamomi ga yin amfani da magunguna
A wasu lokuta, magani iya nuna "Pentas" (Allunan)? Guest masana sun ce da miyagun ƙwayoyi aikin da kyau a lokacin da:
- ulcerative colitis.
- Crohn ta cuta.
Haramta yin amfani da miyagun ƙwayoyi
A karkashin abin da yanayi ba zai iya yin amfani da wani kayan aiki irin su "Pentas"? Umurnai (Allunan, kuma wasu siffofin da kwayoyi da wannan contraindications) ya ce da wadannan haramci:
- hemorrhagic diathesis.
- jini cututtuka.
- lactation.
- Narkewa kamar fili ulcers.
- na karshe 2-5 makonni na ciki.
- rashin glucose-6-phosphate dehydrogenase.
- da shekaru biyu.
- tsanani na koda gazawar.
- hypersensitivity zuwa jamiái abubuwa.
- mai tsanani hanta insufficiency.
Special kula kamata a yi la'akari da wani magani amfani da farko trimester ciki, kazalika da hanta da koda gazawar.
Medicament "Pentas": umarnin don amfani da
Zabi sashi nau'i na da miyagun ƙwayoyi dogara a kan sarrafawa daga cikin manyan pathologic tsari, kazalika da tsawon na hanji raunuka.
Suppositories "pentasil" da kuma dakatar da aka gudanar a distal siffofin da cutar (proctosigmoiditis). A lokaci guda uku kyandirori amfani a ranar 500 MG.
Yadda za a rubũta baka magani "Pentas" (Allunan)? Umurnai na amfani furta cewa, irin wannan magani yana da shawarar kawai ga kowa siffofin cuta. Ga masu rigakafin dakwai, komowan cutar a Crohn ta cuta da medicament ne amfani sau hudu a rana (1 g mesalazine). Game da rigakafin cutar ta koma dawowa daga UC, a wannan yanayin, da miyagun ƙwayoyi An wajabta sau uku a rana 500 MG.
A wani exacerbation da cutar hanya na lura kamata šauki 8-12 makonni. A lokaci guda kowace rana kamata dauki 400-800 MG na da miyagun ƙwayoyi (sau uku kullum).
A tsanani cuta na iya kara kullum sashi na 3-4 g
Allunan "pentasil" ya kamata zai fi dacewa a dauka kai tsaye bayan wani abinci, ruwa ya matse talakawa ruwa.
Ayyuka da-hali
A wasu lokuta, da miyagun ƙwayoyi a tambaya ne da wadannan illa:
- stomatitis, tremor na wata gabar jiki, bushe baki, juwa ko jiri, tashin zuciya, tawayar yanayi.
- asarar ci, jin palpitations, ƙwannafi, shortness na numfashi a lokacin jiki aiki da amai.
- hematuria, zawo ciwo, tachycardia, hepatitis, ciwon kirji.
- kara hanta enzymes, jini da hawa da sauka, pancreatitis, polyneuropathy.
- crystalluria, tinnitus, proteinuria (furotin tukar tumbi), migraine ciwon kai.
- oliguria, leukopenia, anuria (babu urination), thrombocytopenia, samuwar nephrotic ciwo .
- hypoprothrombinemia, agranulocytosis, eosinophilia, anemia.
Ya kamata kuma a lura da cewa, ci na wannan magani a cikin haƙuri za a iya lura: olisgospermiya, alopecia, photosensitivity, mãsu rauni a wata gabar jiki, lupus-kamar ciwo, rage samar da lachrymal ruwa, parotitis.
Yawan abin sama da kwayoyi
Yawan abin sama da alaka da wajen motsa jiki da karin sleepiness, tashin zuciya, gastralgia, amai da rauni a ko'ina cikin jiki. Don kawar da wadannan cututtuka bukatar m ciki lavage kazalika da nada laxatives magunguna da kuma posindromnoy far.
miyagun ƙwayoyi interactions
A medicament "pentasil" shi ne iya rage cikin kudi na sha na cyanocobalamin. Mesalazine kuma qara da yadda ya dace da uricosuric jamiái (ciki har da blockers na tubular mugunya).
Ya kamata mu ma lura da cewa aiki miyagun ƙwayoyi ƙaruwa ulzerogennosti glucocorticosteroids rage sakamako na rifampicin da kuma kara habaka da yawan guba na methotrexate exerts hypoglycemic sakamako a kan sulfonylurea Kalam, spironolactone, furosemide da kuma sulfonamides.
Specific bayanai
A m na wata guda kashi na mesalazine shi ne shawarar ka dauke shi tare da wadannan ko a sosai kusa da nan gaba. Idan aka bata 'yan allurai, ya kamata ka nan da nan tuntubar likita. An haramta wa daina jiyya a kan nasu.
Wani lokaci baya na rahoto jamiái a marasa lafiya lura fitsari tabo da kuma lambar sadarwa ruwan tabarau a yellow-orange ya dafa.
A lura da mesalazine bukatar m likita dubawa a kan aikin koda tsarin na wani haƙuri. Har ila yau, bincike na haƙuri da fitsari da kuma jini ya zama kai a kai (cikin shakka daga far, kazalika da bayan ta kammala).
Yiwuwar faru na illa a cikin halayen da marasa lafiya da samun wannan magani aka ƙara a wadanda suke "m acetylators".
Tare da ci gaban da m ciwo na rashin ha} uri ga aiki sashi shiri "Pentas" nan da nan ya birkice.
Similar kwayoyi da kuma mabukaci reviews
Shin kana da masaniyar abin da za a iya dauke su maye gurbin magani? A wannan dole ne ka sanar da halartar likita. Kamar yadda wani janar mulki, to analogues na wannan kayan aiki hada da wadannan kwayoyi: "Mesakol", "Salozinal" "Salofalk", "Mezavant", "Mesalazin" "Asacol".
Abin da mutane suke cewa game da wannan kayan aiki, saye? A cewar su martani, ya ce medicament ne mai matuƙar tasiri miyagun ƙwayoyi da cewa za a iya saya a wani kantin magani. Marasa lafiya suna da'awar cewa mesalazine ne sosai kyau bayyana kanta ba kawai a magani amma kuma a cikin rigakafin Crohn ta cuta da kuma ulcerative colitis.
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