Kiwon lafiya, Shirye-shirye
Da miyagun ƙwayoyi "Chlorpromazine": reviews na likitoci, umarnin don amfani, abun da ke ciki da kuma bayanin
Antipsychotic kwayoyi - mai psychotropic kwayoyi, wanda aka tsara domin lura da psychotic cuta. Ya kamata a lura da cewa gargajiya sunan wannan kwayoyi - neuroleptics. Wadannan kwayoyi iya yadda ya kamata tasiri cikin cututtuka kamar masifa, ainihin komai bane illa kawayeniya, hallucinations, ya zaci rashin lafiya, psychotic agitation, hali cuta , da sauransu. D. Sanya wadannan kwayoyi za a iya samu likita.
Mafi mashahuri antipsychotic miyagun ƙwayoyi abubuwa "Chlorpromazine". Umarnin don amfani, price, reviews, analogs, Contra-alamomi da miyagun ƙwayoyi aka gabatar a kasa.
Abun da ke ciki, description, fom
Abin da nau'i ne muhimmi a da miyagun ƙwayoyi "Chlorpromazine"? Umurnai, reviews bayar da rahoton cewa wannan magani ne aka sayar a cikin nau'i na brownish-m kwayoyi, kazalika da wani bayani ga igiyar jini da kuma intramuscular gwamnati. The aiki abu na nufin bayanan ne chlorpromazine hydrochloride. Har ila yau, dangane da saki form su dauke da dama extras.
pharmacological siffofin
Mene ne na ƙwarai miyagun ƙwayoyi "Chlorpromazine"? Umarnin don amfani, martani nuna cewa wannan shi ne wani antipsychotic wakili, wanda ta pharmacological kungiyar tana nufin neuroleptics. Yana yana da wani hypotensive, antiemetic da antihistamine effects.
The aiki sashi na wannan miyagun ƙwayoyi ne a wanda aka samu daga phenothiazine. Bugu da kari a wadannan kaddarorin aiki medicament mallaka magani mai kantad da hankali, hypothermic rauni, antipsychotic, gida irritating, vasodilating da moderately M-anticholinergic effects.
Antipsychotic sakamako daga cikin kayan aiki da ake samu ta hanyar tarewa dopamine D 2 rabe da mesolimbic tsarin Mesocortical. Saboda irin kaddarorin da miyagun ƙwayoyi ne iya kawar hallucinations, r ?? i kuma sauran m bayyanar cututtuka na psychosis.
Ya kamata a lura kuma cewa "Chlorpromazine", reviews na wanda aka jera a kasa, sauqaqa daban-daban iri psychomotor agitation, mutunci da kuma rage tsanani daga psychotic tsoro.
Magani mai kantad da hankali sakamako daga cikin miyagun ƙwayoyi aka samu da tarewa da adrenergic reticular kantin cewa suna located a cikin brainstem.
Properties na da miyagun ƙwayoyi
Mene ne Properties muhimmi a cikin medicament "Chlorpromazine"? Reviews sun ruwaito cewa wannan magani mai depressing sakamako a kan sharadi reflex aiki, hūta kwarangwal tsokoki, da rage maras wata-wata mota aiki, rage ji na ƙwarai to na ciki da kuma exogenous samuwar kasashe da wani kwari hankali. A amfani da manyan allurai da miyagun ƙwayoyi sa mai tsanani drowsiness.
Kawancen na vagus jijiya a cikin gastrointestinal fili da kuma dopamine D2 rabe dake a cikin emetic jawo zone da cibiyar samar da antiemetic sakamako daga cikin miyagun ƙwayoyi. Ya kamata kuma a lura cewa wannan makaman da kadan sakamako a kan M-cholinergic rabe. Bugu da ƙari, ta furta sakamako lura ga alpha-adrenergic rabe.
A mataki na miyagun ƙwayoyi
miyagun ƙwayoyi "Chlorpromazine" Yaya ta yi aiki? Reviews ce cewa wannan kayan aiki ne iya gaba daya kawar da effects da aka sa ta epinephrine. Its hypothermic effects saboda kawancen na dopamine rabe cewa suna located a cikin hypothalamus.
An fito da miyagun ƙwayoyi lowers jini, zuciya rate ƙaruwa, yana mai rauni antihistaminic sakamako da kuma bayyana kataleptogennoe mataki, da kuma rage permeability na capillary katangu.
Domin intramuscular gwamnati da medicament sa kwantad da hankali a lokacin ¼ hours, da kuma bayan baka gwamnati - bayan 120 minti. Haƙuri haƙuri ga magani mai kantad da hankali da kuma hypotensive sakamako tasowa a game da mako guda.
Lokacin da ka karɓi wannan magani a cikin ya antipsychotic kaddarorin da wani sakamako a kan 4th ko 7th rana. A warkewa sakamako daga cikin miyagun ƙwayoyi yana game 2-6 watanni.
A pharmacokinetics da miyagun ƙwayoyi
Shin, "Chlorpromazine" sucked? Reviews rahoton cewa an baki chlorpromazine azumi amma ba gaba daya tunawa daga narkewa kamar tsarin. Its ganiya jini yawa samu bayan 4 h.
Wannan magani shigarsu farko ratsa cikin hanta. Saboda haka ta maida hankali a cikin jini bayan baka gwamnati ne sosai kasa da maida hankali bayan intramuscular gwamnati.
Da miyagun ƙwayoyi ne metabolized a cikin hanta to m da kuma aiki Kalam.
Chlorpromazine yana da babban bond to jini sunadaran. An yadu rarraba a jikin haƙuri, iya shiga ta hanyar da BBB.
Half-rai na aiki abubuwa na miyagun ƙwayoyi ne game da minti 30. Kamar wancan ne kawar da Irinta iya zama ya fi tsayi.
Nuna medicament dauke tare da fitsari da kuma bile.
Drug "Chlorpromazine": alamomi ga yin amfani da
Reviews sun ruwaito cewa da miyagun ƙwayoyi ne yadu amfani a cikin tabin hankali yi. Kuma an wajabta, a lura da agitation a mutumin da schizophrenia. Har ila yau, wannan magani da ake amfani a kullum psychosis, m delusional jihohi, hypomanic tashin hankali, rashin barci, psychopathy, shafi tunanin mutum rashin lafiya, tashin hankali, tsoro da tashin hankali.
Bugu da kari a yanayi da aka lissafa alamomi ga yin amfani da wannan magani ne: m hiccups, giya psychosis, wanda ba a iya lura da shi ba amai da kuma mai tsanani tashin zuciya. Idan akwai zafi da miyagun ƙwayoyi kara habaka sakamakon analgesics.
Ya kamata kuma a lura da cewa, nufin sanya gani a cututtuka wanda suna tare da ƙara murdede sautin, tetanus (as hade far a tare da tare da barbiturates) da kuma bayan daban-daban disturbances a cerebral wurare dabam dabam.
Ba haka ba da dadewa, wannan magani da ake amfani da wucin gadi hypothermia hada lytic garwayayye. A anesthesiology wannan magani sau da yawa wajabta kwantad da hankali da kuma janar maganin sa barci potentiation.
A dermatological yi "Chlorpromazine" (martani da marasa lafiya game da miyagun ƙwayoyi ne yafi kyau hali) a yi amfani da itching dermatoses. Bugu da kari, shi za a iya amfani da magani daga m porphyria hali.
contraindications
A wasu lokuta, ba wajabta antipsychotic "Chlorpromazine"? Reviews likitoci bayar da rahoton cewa wannan kayan aiki ba a yi amfani da comatose jihohin daga duk wani tushen, kazalika a marasa lafiya tare da tsanani da zalunci da juyayi tsarin, mai tsanani cututtukan zuciya da kuma jijiyoyin bugun gini rashin ha} uri ga aiki abu, wani m cuta na kwakwalwa da kuma kashin baya na tsari yanayi na kwakwalwa, ulcerative raunuka na gastrointestinal fili da kuma a lokacin da nono ciyar.
A ra'ayi na babban hadarin da hepatotoxic halayen, yana nufin wajabta tare da matsananci hankali a shan barasa. A wannan gaskiya ne daga nono, da jini dyscrasias, hyperplasia na prostate gland shine yake, glaucoma, rufe-nau'i, Parkinson ta cuta, epilepsy, myxedema, amai, cachexia, Reye ciwo da kuma tsofaffi.
Drug "Chlorpromazine": umarnin don amfani da
Allunan ratings wanda aka gabatar a nan, a yi amfani da tabin hankali yi a fara kullum sashi daidai 25-100 MG. Wannan adadin ne zuwa kashi 1-4 allurai. A tsawon lokaci, kara da kashi kowane kwanaki hudu ga 25 ko 50 MG ga cimma da ake so sakamako.
Tare da tashin hankali preoperatively aiki miyagun ƙwayoyi sha for 2-3 hours.
A kalla guda kashi na wannan wakili ne 300 MG, da kuma kullum - 1,5 g
Game da bayani, shi ne gudanar intravenously ko intramuscularly. Harufan sashi na wannan magani ne 25-50 MG.
Kafin gwamnatin da miyagun ƙwayoyi da shi da aka diluted da 2.5 ml na sodium chloride bayani ko procaine. Injections yi zurfi intramuscular allura.
A kalla guda kashi na wannan wakili ne 150 MG da kullum - 1 g As for igiyar jini gwamnati, wadannan dabi'u dace 100 da kuma 250 MG.
a ke so effects
Haddasa wani gefen effects "Chlorpromazine" (Allunan)? Reviews sun ruwaito cewa farkon matakai na lura da wannan magani zai iya sa bushe baki, paresis na masauki, frigidity, ta ƙara drowsiness, maƙarƙashiya, barci cuta, juwa ko jiri, illa ci, tachycardia, ya nuna wani nau'i na orthostatic hypotension, urinary riƙewa, rage iko, alerji da fall jini.
Tsawo far tare da wannan magani yana sa tsoka cramps wuyansa, kuma harshe, neuroleptic ciki Akinetes-m sabon abu, extrapyramidal cuta, amenorrhea, akathisia, jinkiri dauki zuwa daban-daban samuwar kasashe, hypercoagulability, amai, shafi tunanin mutum da canje-canje, cardiac arrhythmia, pigmentation na fata, hanawa na bargo hematopoiesis , gynecomastia, cholestatic jaundice, galactorrhea, giperplolaktinemiyu, oliguria, zawo, da kuma neuroleptic m ciwo. Tare da igiyar jini jiko phlebitis kafa da intramuscular - infiltrates.
takamaiman shawarwari
Far da wannan kayan aiki na bukatar mai da hankali iko da jini, bugun jini, aiki da kodan da kuma hanta.
Wannan magani zai iya sa photosensitivity, sabili da haka a lokacin da ya m bada shawarar don kauce wa fiddawa.
Analogs da kudin
Farashin wannan magani dogara a kan saki form. Marufi da 10 vials za a iya saya don 60 rubles, yayin da a irin wannan yawan Allunan ne game da 150 rubles.
By analogues wannan magani hada da "Chlorpromazine hydrochloride" da "Tisercinum".
reviews
A cewar masana dauke da medicament yana da m antipsychotic sakamako, cire duk alamun psychomotor agitation. Duk da haka, ya kamata a lura da cewa wannan na nufin sake dubawa ne na daban-daban yanayi.
Wasu marasa lafiya da cewa wannan magani ne tasiri a Alzheimer ta cuta, schizophrenia, psychosis, epilepsy, da kuma wani da-sauqaqa tashin hankali da danniya. Wasu da masu amfani da imani cewa dauke magani tsokani ci gaban da farfadiya seizures, hannunka-shake, daban-daban hali cuta da kuma wuce kima sleepiness jihar.
A cikin wani hali, wannan magani ya kamata kawai a yi amfani a matsayin nufi da a karkashin kulawa da halartar likita.
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