Kiwon lafiyaShirye-shirye

"Teopeka" (300 MG): umarnin don amfani, alamomi, manufacturer

Mutane da asma, ya san yadda muhimmanci lokaci don taimaka tare da bronchospasm. Wani lokaci daidai mataki a cikin wannan halin ba zai iya ceton rayuka. A muhimmiyar rawa a samun mutane daga huhu matsaloli wasa bronchodilators.

Description of shiri

"Teopeka" (300 MG), da umarnin don yin amfani da abin da aka nuna a cikin wannan takarda shi ne wani farin Allunan ploskotsilindricheskoy madauwari siffar, wanda ake cushe a shiryawa kwane-kwane. Babban aiki sashi daga cikin miyagun ƙwayoyi ne theophylline. Its taro a guda kwamfutar hannu na shirye-shiryen da wannan nau'i ne 300 MG.

Ta yaya wannan magani?

By ta pharmacological mataki na theophylline, wanda yake shi ne wanda aka samu daga purine, yana da wani inhibiting sakamako a kan phosphodiesterase. The aiki sashi daga cikin miyagun ƙwayoyi tubalan da takamaiman purine rabe, stimulates Camp jari a nama depots, lowers da ikon da m tsoka nama mu'ãmalar, rage adadin free alli ions, wanda ƙaura ta hanyar cell membranes.

Alama furta vasodilating sakamako liyafar "teopeka" shiri (300 MG). Umurnai na amfani bayyana dukiya a matsayin wani tasiri a gefe jini. Theophylline qara jini ya kwarara ta cikin koda tsarin, da inganta harkokin shakatawa na Bronchial m tsoka da jini. Har ila yau, da mataki na aiki bangaren ne halin da m diuretic. Theophylline ya hana a saki abubuwa da fita, ya sa wani rashin lafiyan martani kazalika qara da zaman lafiyar na mast cell membranes. Idan wani m hypokalemia aiki abu intensifies iska.

Theophylline taimaka normalize aiki na numfashi, kunna daidai cibiyar a cikin kwakwalwa, sakamakon shi a mafi jini oxygen jikewa, shi rage-rage na maida hankali ne carbon dioxide. Drug "teopeka" stimulates diaphragm, suna ɓuɓɓugar da shi yanka. Yana kuma qara da darajar da nuna alama na mucociliary yarda aiki intensifies numfashi da kuma intercostal tsokoki.

Theophylline take kaiwa zuwa al'ada jini mikrotsirkullyatsiyu rage thrombus samuwar, musamman factor cike da gusar tari na platelet Kwayoyin. miyagun ƙwayoyi kuma inganta da ya kwarara daga jini quality, qara jure deforming erythrocytes dalilai.

"Teopeka" (300 MG), game da shi, rage total matsa lamba a cikin huhu wurare dabam dabam, da kuma rage juriya a cikin huhu jijiyoyin bugun gini tsarin. A sakamakon haka, da sautin da fata integuments, koda da kwakwalwa da rage-rage. A sakamakon samun theophylline alama ruri na jijiyoyin zuciya jini ya kwarara, ta ƙara cardiac aiki, karuwa da tsokar mai ban mamaki Kwayoyin bukatar oxygen, har ya rãyar da bugun jini, da ƙarfin zuciya contractions karu.

Pharmacokinetics da pharmacodynamics da miyagun ƙwayoyi

Bayan da haƙuri dauki kwaya da theophylline, da abu an tunawa daga cikin gastrointestinal fili. Abinci sha yana da wani sakamako a kan kudi na sha na da miyagun ƙwayoyi, amma mataki na sha da kuma yarda ya zauna canzawa. Tun da jini da furotin da ta ɗaure 40% na aiki abu. Theophylline metabolism auku a cikin hanta da cytochrome P450.

Tukar tumbi da metabolites samar a cikin aiki nau'i via kodan, amma 10% daga cikin miyagun ƙwayoyi ne shafe a asalin siffan. Wasu dalilai da wani gagarumin sakamako a kan metabolism na theophylline. Smoking, shan wasu magunguna, abin da ake ci halaye, comorbidities, shekaru, iya sa sabawa musayar daga cikin aiki dũkiyõyinsu a cikin jikin mutum. Rage yarda da theophylline aka lura a huhu edema, cutar hanta, COPD, kuma a zuciya rashin cin nasara.

Wa zai iya yi maraba da wannan kayan aiki?

Akwai wasu yanayi na wanda wani "teopeka" (300 MG). Umurnai na amfani bayyana da wadannan cututtuka:

  • obstructive mashako a kullum form.
  • barci apnea.
  • emphysema.
  • asma.
  • na huhu hauhawar jini.
  • na huhu zuciya.

Har ila yau, da miyagun ƙwayoyi "teopeka" tabbatacce feedback wanda za a iya amfani a tare da tare da sauran kwayoyi da magani daga koda edema yanayi. Marasa lafiya lura da high dace na kayan aiki da kuma ta karbar domin lura da cututtuka na numfashi tsarin.

contraindications

Duk da haka, wannan magani za a iya amfani da ba kowa da kowa, saboda na kasancewar wani adadin da gargadin da kudi. "Teopeka" contraindications ne kamar haka:

  • hemorrhagic bugun jini irin;
  • epilepsy.
  • zub da jini daga gastrointestinal fili a tarihi.
  • miki samuwar a cikin narkewa kamar gabobin.
  • tachycardia high severities.
  • hauhawar jini ko hypotension.
  • hypersensitivity.
  • gastritis, tare da high acidity.
  • Yara har zuwa shekaru 12 years.

A gaban akalla daya daga wadannan syndromes ko yanayin da miyagun ƙwayoyi theophylline kamata bari

illa

Akwai quite wani babban rukuni na gefe-effects daga shan "teopeka" shiri (300 MG). Umurnai na yin amfani da su da hannun jari a kan tsari bayyananen:

  • cuta na juyayi tsarin: ciwon kai, dizziness, barci disturbances, restlessness, ta ƙara tashin hankali da kuma irritability, tremors.
  • tabarbarewa na zuciya da jini: tachycardia, arrhythmia, hypotension, ta ƙara mita na angina harin, ƙarya angina.
  • take hakkin gastrointestinal al'ada aiki: tashin zuciya, gastralgia, amai, ƙwannafi, reflux, exacerbation ulcers, zawo, rage ci.
  • bayyananen na rashin lafiyan halayen: fata rash, zazzabi, itching.
  • tsakanin sauran m events daga shan miyagun ƙwayoyi aka lura: tachypnea, albuminuria, ta ƙara diuresis, zafi a cikin sternum, hematuria, flushing, ta ƙara sweating, gipoglekemiya.

Yawanci, da gyara da kashi don rage illa an rage ko ceases gaba ɗaya.

Yadda za a yi da miyagun ƙwayoyi?

Yana nufin daga mashako, kamar "teopeka" an sanya kawai da halartar likita da su sashi ne aka zaba a kan wani mutum akai. A talakawan kullum Nome karkacewa 400 MG theophylline. Idan wani m daukawa da miyagun ƙwayoyi da kyau, to bayan kwanaki 2-3 daga farko kashi na magani, da ƙarfi ya karu da 25% da kuma kara da likita ta hankali.

A kan samun nufin daga mashako "teopeka" a kullum kashi na kasa da 900 MG theophylline ciki iko ba lallai ba ne a cikin haƙuri na jini. Idan ka duba bayyanuwar maye, da gaggawa bukatar kafa iko a kan matakin da taro na babban aiki sashi a cikin jini. Mafi dauke Manuniya 10-20 micrograms da ml. Idan theophylline abun ciki na haƙuri da jini ne mafi girma fiye da na al'ada, da kiyaye ci gaban korau halayen. A wannan yanayin wajibi ne don rage sashi daga cikin miyagun ƙwayoyi, da kuma a warkewa sakamako zai raunana.

Shin akwai wani yawan abin sama?

Bronchodilators kamar "teopeka" na iya haifar da tsanani da cuta na jiki a taron na yawan abin sama. Lokacin da yadda ya kamata ya dace kullum kudi na samun wajen da wadannan cututtuka zai iya bayyana:

  • rage ci.
  • rashin barci.
  • zawo.
  • na ramin zuciya arrhythmias siffar.
  • tachycardia.
  • zub da jini na narkewa kamar tsarin.
  • tachypnea.
  • tsãwa;
  • tashin hankali.
  • yankin Flushing da fata .
  • ya karu excitability.
  • tsoro da haske.
  • amai jini.

Yana kuma iya ci gaba mai tsanani da guba, wanda bayyana kanta a cikin wadannan cututtuka:

  • abin da ya faru na farfadiya seizures.
  • hypokalemia.
  • koda gazawar, myoglobinuria.
  • hypotension.
  • rikice.
  • hyperglycemia.
  • rayuwa acidosis.

Abin da ya yi a cikin wannan hali?

Idan akwai shaida daga ãyõyi, ko tuhuma da su bukatar yin ciki lavage, ba da haƙuri chelators, laxatives, kwayoyi, kazalika da shirya diuresis plasmasorption, hemodialysis da hemosorption. Idan haƙuri ne da ciwon seizures, to, shi ne shawarar gabatar da oxygen far da kuma igiyar jini "Diazepam" cewa za ta taimaka yadda ya kamata tsara kãmun. A cikin hali na furta tashin zuciya da kuma amai ya sanya igiyar jini "Ondansetron" kwayoyi da kuma "Metaklopromida".

Abin da magunguna ba za a iya hada "teopeka"?

Bronchodilators kamar "teopeka 'kada kai tare da wani macrolide-kwayoyin" Allopurinol "," cimetidine "," Lincomycin "," isoprenaline ", kazalika da na baka hana saboda wadannan kwayoyi taimaka wajen rage yarda da theophylline.

An ba da shawarar hada ci daga beta-blockers, musamman wadanda ba zabe, tare da miyagun ƙwayoyi "teopeka", daga abin da zai iya ci gaba Bronchial constriction da rage bronchodilator sakamako na theophylline.

Idan "teopeka" amfani tare da "Furosemide" maganin kafeyin da sauran abubuwa da ta da beta-2 adrenergic rabe, da ayyukan da ta farko bangaren da aka muhimmanci karu. Idan hade tare theophylline "Aminoglutitemidom", na farko abu fara rayayye excreted daga jiki da kuma ta yadda ya dace saukad.

"Acyclovir" shi ne iya kara maida hankali ne babban aiki sashi "teopeka" kuma qara illar da ta liyafar. Similar mamaki ne kiyaye a lokacin da co-gudanar da theophylline kwayoyi "Dialteazem", "Felodipine" "Verapamil", "Nefedipin". Wadannan magunguna ba su canja bronchodilator sakamako, duk da haka, haƙuri iya samun bayyanar cututtuka na m halayen ko yawan abin sama.

Abu "Disulfiram" iya kara theophylline jini to m Manuniya m mai guba rauni. "Propranolol", da bambanci, rage "teopeka" yarda da aiki abu. Taro na theophylline an karu da somestnom ta liyafar tare da "enoxacin" da kuma fluoroquinolones. Lokacin da theophylline far rage-rage yadda ya dace da lithium salts.

Idan hada magani tare da "pentobarbital", "Carbamazepine", "Isoniazid", "rifamycins", "sulfinpyrazone" ƙãra yarda "teopeka" da kuma rage ingancinta. Lokacin da concomitantly da theophylline "phenytoin" akwai juna hanawa na aiki bangaren a cikin haƙuri na jini.

Waɗannan jagororin suna da muhimmanci musamman, kyalewa su ne fraught tare da kiwon lafiya da matsaloli. Saboda haka, kafin shan "teopeka", karanta umarnin a hankali. Kuma idan kun ake jinyar ga wani na sama magunguna, tuntuɓi likita.

Yadda za a saya da miyagun ƙwayoyi da kuma yadda da miyagun ƙwayoyi ne da daraja?

A ra'ayi na tsanani contraindications da kuma gefen sakamakon wannan miyagun ƙwayoyi, "teopeka" saki a Pharmacy kawai ta sayen magani.

Drug "teopeka" Farashin ne da talakawan a Rasha ne 160 rubles, gabatar a Pharmacy da daban-daban masana'antun. Daya jinsunan - magani ga "Borschagovsky CPP SPC" Ukrainian pharmaceutical kamfanonin. Its kudin ne 155 rubles. Rasha samar da "teopeka" miyagun ƙwayoyi, 300 MG ne da za'ayi a cikin kamfannoni na JSC "Pharmaceutical kasuwanci" da "Valens". wadannan kwayoyi kudin 290 rubles da 190 rubles bi da bi.

A general, da miyagun ƙwayoyi "teopeka", Farashin ne m, dauke araha magani domin da yawa daga cikin 'yan ƙasa. A kwatanta da Turai da takwarorinsu da wannan kayan aiki ne da yawa mai rahusa. Rasha samar da "teopeka" da miyagun ƙwayoyi sanya shi araha.

Tsõratar da lokacin shan magani

Lokacin da samun "teopeka" miyagun ƙwayoyi, da sake dubawa na waxanda suke da kyau, ya kamata kula da wadannan bayanai. Idan haƙuri yana da jijiyoyin zuciya ko cardiac insufficiency, atherosclerosis, cardiomyopathy, gastrointestinal miki, cutar hanta, prostate ciwon daji, oesophageal reflux, ciki, hypothyroidism ko ya karu propensity zuwa seizures, da miyagun ƙwayoyi theophylline ya kamata a dauka tare da taka tsantsan.

Yara a karkashin shekaru 12 da haihuwa da kuma mazan marasa lafiya "teopeka" nada wuya.

Zai yiwu amfani da rectal siffofin da miyagun ƙwayoyi, amma da suka kamata a yi amfani matsa a hankali a pathologies daga cikin dubura da kuma zawo ciwo. Marasa lafiya da jaraba ga shan taba maki ragewan sakamako na lura "teopeka".

Dauke inadmissible hadin gwiwa magani theophylline da xanthine Kalam. Idan haƙuri ne tsofaffi ya bayyana concomitant cututtuka, kwayar cutar, cutar hanta, zuciya da jini, likita wajibi ne don gyara kashi na magani.

Zan iya daukar wani magani ga mata masu ciki?

A ciki mace da medicament an nuna for gaban tsanani alamomi tun theophylline ne iya shiga cikin mahaifa. Idan liyafar "teopeka" ya nuna shayar da mama, da lactation ya kamata a katse.

Wannan manual ne a Saukake version na cikakken umarnin, wanda aka haɗe da miyagun ƙwayoyi "teopeka". Ya kamata a karanta a hankali kafin amfani da shi. Idan akwai wani abu da kake rude ko a cikin shakka, tuntuɓi likita.

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