Kiwon lafiyaShirye-shirye

Drug "Sotageksal", analogs da feedback a kan su

Arrhythmia - shi ne mai irin zuciya rate, wanda shi ne daban-daban daga al'ada sinus kari. Lokacin da arrhythmias a cikin mutane akwai daya ko dama keta zuciya. A Pathology iya gabatar a matsayin mita da kuma ikon karawa zuciya rate (tachycardia) da kuma, conversely, da rage a su (bradycardia). Katsalandan ga aikin zuciya tsoka, kuma suna a wani m mutum. Duk da haka, a mafi yawan lokuta, da arrhythmia ne a tare da sauran cardiac cututtuka. Irin wannan jiha ne m, a cewa ya karu excitability na zuciya tsoka - myocardium, wanda zai iya kai ƙarshe zuwa zuciya rashin cin nasara idan ya bar untreated.

akwai shirye na musamman domin daidaita zuciya rate, daya daga wanda yake shi ne "Sotageksal". Analogues da miyagun ƙwayoyi ne ma yadu a yi amfani likita yi. Wadannan kwayoyi ne zuwa rukuni na magunguna da cewa suna da antiarrhythmic ayyuka, da kuma beta-blockers. Lokacin da ingested, suka toshe beta-adrenergic rabe, wanda aka located a cikin m tsoka, cardiac tsoka da sauran tsokoki, da kuma ke da alhakin jiki ta mayar da martani ga alãmõmin danniya. Overall kardioeffekt ne don rage mita da kuma tsanani da zuciya kudi, da rage-rage cardiac madugu. Kamar yadda wani tsari sakamako ne ma ya lura ragewan na jini matsa lamba a kan ganuwar da jijiyoyin zuciya tasoshin.

da miyagun ƙwayoyi

"Sotalol» (Sotalol) - rene ta kasa da kasa sunan a duniya da miyagun ƙwayoyi "Sotageksal". Analogs na abun da ke ciki na iya samun wani daban-daban, amma irin wannan antiarrhythmic sakamako. Babban aiki abu "Sotageksal" ya ƙunshi sotalol hydrochloride. Bugu da kari, shi ya hada da wani karamin yawan karin aka gyara. Daga gare su, - cellulose, lactose monohydrate, masara sitaci, magnesium stearate da sauran binders.

A shiryayye rayuwar Allunan, ko injectable bayani ne shekaru 5.

"Sotageksal" analogues da kuma abun da ke ciki

Daya kwamfutar hannu na wannan samfurin ya ƙunshi 40, 80 ko 160 MG na aiki abu. An samar da yafi a matsayin White zagaye Allunan da daya gefen dan kadan convex kuma embossed tare da raguwa SOT. A baya na kwamfutar hannu da aka bisected ta wajen dosing domin saukaka wa kasada. All cushe a blisters na 10 guda, kuma kwali kwalaye. Kowane cuta iya Range daga 1 zuwa 10 blisters (na daga 10 zuwa 100 guda na alluna).

Har ila yau, "Sotageksal" da aka samar a cikin nau'i na bayani ga igiyar jini allura. Kowane ampoule ƙunshi 4 ml da miyagun ƙwayoyi. A 1 ml na bayani ne 10 MG na tsarki na asali abu. A miyagun ƙwayoyi ya kamata a kiyaye shi daga hasken rana duhu da kuma bushe wuri, a cikin abin da yara da damar yana da iyaka.

Analogs tare da aiki abu sotalol hydrochloride Allunan kerarre:

  • "Sotaleks" (160 MG).
  • "Soritmik" (ta 0,16 g).
  • "Sotalol Canon" (80 da 160 MG).
  • "Darob" (80 da 160 MG).
  • "Tenzol" (80 da 160 MG).

pharmacological effects

"Sotageksal" analogues da ma'ana da miyagun ƙwayoyi da pronounced anti-arrhythmic sakamako. Wannan aka samu da nagarta na da ikon toshe β-adrenergic rabe da kuma hana potassium tashoshi. Kwayoyi kara tsawon lokacin hatsaisai da reflex lokaci atria da ventricles. Kara da sautin na Bronchial m tsoka da tsoka Layer da jirgin ruwa katangu. Rage tsokar contractility.

Sotalol hydrochloride yana da wani dukan sa na Properties. Yana da wani mummunan chronotropic, dromotropic, batmotroponoe da inotropic sakamako na Jamus miyagun ƙwayoyi "Sotageksal". Analogs, da abun da ke ciki na wanda shi ne m, na iya samun wani iri sunan. Su ma iya rage zuciya kudi da kuma su iko. Saboda wannan bukatar tsokar oxygen amfani ne ƙwarai rage. Kuma a sakamakon, da kaya a kan zuciya ne rage.

Absorption da tukar tumbi da kwayoyi

Drug sha ne m. Its bioavailability ne 90%, da kuma sha - game da 80%. A cikin 2.5-4 hours of matsakaicin maida hankali na aiki sashi aka samu bayan karbar jini. Bayan igiyar jini gwamnati, da sakamako ne riga da ya bayyana bayan 5-10 minti. Absorption auku a 20% mafi alheri, kuma sauri idan ka dauki magani kan komai a ciki. Saboda gaskiya cewa solubility na dũkiyõyinsu a cikin fats ne ragu, sotalol hydrochloride ba za a dauka a lokaci guda tare da kiwo kayayyakin da fats na dabba da asali.

Ba tare da ake daure wa jini sunadarai, da miyagun ƙwayoyi ne rarraba a cikin tsokoki da kuma na gefe gabobin ko'ina cikin 3-4 kwanaki na yau da kullum m. A lokaci guda, da kuma shi cimma wani tabbatacce sakamako a kan hauhawar jini. A cerebrospinal ruwa da miyagun ƙwayoyi maida hankali ne ba fiye da 20%. Action bayan allura ya ci gaba har zuwa 2 hours. sakamako ta ci gaba bayan baka dosing na alluna "Sotageksal" to 12 hours. Analogs da miyagun ƙwayoyi a cikin abun da ke ciki wanda ya ƙunshi sotalol hydrochloride, kuma ba mai saukin kamuwa zuwa metabolism da kodan da excreted a cikin fitsari (90%) kuma tumbi a kan talakawan cikin 10-20 hours.

Wannan shi ne dalilin da ya sa marasa lafiya da illa na koda da kuma urinary tsarin ya nuna da magani zuwa karami sashi. Mazan mutane sukan lura da shekaru da alaka da tabarbarewar koda aiki. Wannan na taimaka wa gaskiya cewa abu ne nuna a hankali kudi da kuma iya tara a cikin jiki. Saboda haka, wannan rukuni na marasa lafiya da miyagun ƙwayoyi a yi amfani da hankali da kuma sashi ne m akayi daban-daban.

A magani taimaka wajen normalize musayar oxygen a cikin tsokoki, da gusar irritability, tashin hankali, danniya da kuma sauran abubuwan da suka shafi da mita da kuma tsanani da contractions daga cikin zuciya.

"Sotageksal": umarnin don amfani da

Analogs da miyagun ƙwayoyi da kuma wakili aka yi amfani da asalin sunan ga symptomatic cardiac arrhythmias, domin lura da na ramin zuciya arrythmia. Amma akwai wani daban-daban sakamako a marasa lafiya tare da kama diagnoses. Saboda haka, dole ne ka sanya wani likita bayan wani na sosai jarrabawa da kuma tsananin a kan shaida.

Qalilan ne wakili amfani da magani na marasa lafiya da suka yi psoriasis (psoriasis) ko wahala daga ciwon sukari da illa carbohydrate metabolism. Zama wary sanya mutanen da suke da wani tarihi na alerji ne ba, yana nufin "Sotageksal". Analogues shi ne ma iya kashe jiki ta ji na ƙwarai to rashin lafiyan samuwar kasashe. Hankali magani da ake amfani da su bi da marasa lafiya da zuciya rashin cin nasara, yiwuwa ga m depressions. Marasa lafiya da suka yi a tsokar zuciya infarction, arrhythmia hadarin kaifafa a lokacin liyafar "Sotageksala".

Sashi da magani lokaci

Dangane da tsanani da cuta ne niyya da kuma tsawon lokaci na miyagun ƙwayoyi far "Sotageksal". Umurnai na amfani (analogs iya samun wasu umarnin ga liyafar) ya ƙunshi da wadannan shawarwari:

  • kwamfutar hannu da aka yi lõma da dukan, ba chewed kuma da yalwa da ruwa.
  • Yanayin aiki aka yi domin 1-2 hours kafin cin abinci.
  • dauki magani 2-3 sau a rana.

Jiyya da wuri kullum kashi kada fi 80 MG (1 kwamfutar hannu) hauhawar jini da kuma tachycardia. Duk da haka, a cikin rashi na so warkewa sakamako kashi karu. A hankali, tare da wani tazara na kwanaki 2-3 shi ne gyara ga 240-320 MG da rana, amma kawai a wani asibiti. A mafi inganci shi ne a hankali a hankali karuwa a sashi na 80 MG da mako.

A kalla kashi iya zama 6 Allunan da rana miyagun ƙwayoyi "Sotageksal". Analogues, da sashi na wanda ƙila za a ƙara idan likita gan shi ya cancanta, za a nada akayi daban-daban. Ko akwai barazana ga rayuwa, jimlar adadin aiki sashi kada wuce 480 MG da rana.

Idan haƙuri ba koda aikin cuta, da jiyya regimen zaba a matsayin aiki na creatinine yarda. Its karuwa (har zuwa 30 MG / min), da kashi ne yawanci rage zuwa guda biyu zuwa sau hudu.

Igiyar jini injections sanya sau biyu a rana, zuwa kashi biyu ampoule allura na 2 ml. The bayani ne allura sannu a hankali a kan 5-7 minti. A lokacin jiyya, da ake buƙata iko da jini, bugun jini, da kodan da kuma urinary tsarin, creatinine yarda a magani.

shaidar

Kudi kaddamarda domin lura da wadannan cututtuka:

  • tachycardia, na ramin zuciya.
  • Wolff - Parkinson - White;
  • cardiomyopathy.
  • na ramin zuciya wanda bai kai lashe.
  • mitral bawul prolapse.
  • Paroxysmal atrial fibrillation da atria.
  • hauhawar jini (hawan jini).
  • rigakafi da magani daga tsokar zuciya infarction (a wasu lokuta).

A tsanani illa koda aiki, wani likita da aka zamar masa dole ya ci gaba da saka idanu da taro na aiki abu a cikin jini magani da kuma daidaita kashi "Sotageksal" miyagun ƙwayoyi. Analogs na alamomi ga m ne m. Amma, duk da wannan, nasu canza daya miyagun ƙwayoyi zuwa wasu ne tsananin haramta. Sokewa magani ya kamata faruwa nan da nan, amma sannu a hankali. Ba zato Tsayawa zai iya sa deterioration na asibiti yanayin.

contraindications

Duk wani antiarrhythmic wakili ba zai iya ko da yaushe a sanya wani haƙuri, ciki har da "Sotageksal". Analogs contraindications ne guda, suka ba za a iya amfani da a karkashin wadannan yanayi:

  • hypersensitivity ko idiosyncrasy asali abu ko wani karin bangaren.
  • rauni sinus kwana.
  • alama raguwa a zuciya rate (bradycardia).
  • kullum obstructive na huhu matakai.
  • m Bronchial fuka.
  • koda gazawar.
  • m tsokar zuciya infarction.
  • m ko na kullum zuciya maye.
  • cardiogenic buga.
  • elongated QT tazara ciwo .
  • yara shekaru.
  • alerji, rashin lafiyan rhinitis.
  • ciki da kuma nono.
  • rage matsa lamba (hypotension).
  • janar maganin sa barci.
  • gangrene.
  • gefe jijiyoyin bugun gini cuta.
  • ci gaban da tachycardia type "pirouette" (yanayin da aka yi fama mafi sau da yawa a cikin mata fiye da a maza).

Isasshen kwarewa tare da miyagun ƙwayoyi a lokacin daukar ciki ba. Kawai "Sotageksal" nada a kan m alamomi. Takwarorinsu a cikin ta farko trimester kuma barazana ga fetal rayuwa, da kuma shan su iya kai ga zubar da ciki. M bincike data a kan m da miyagun ƙwayoyi a mata haihu har yanzu ba shi da.

A karshe watanni na far za a progressively rage for 2-4 kwanaki kafin ceto, idan wata mace ta daukan shi a lokacin da dukan tsawon ciki. Wannan ne yake aikata to tabbatar da cewa jariri ba da zalunci na numfashi ayyuka, bradycardia ko hypotension saboda da miyagun ƙwayoyi "Sotageksal".

Analogues dangane sotalol hydrochloride ya kamata a daina amfani da su dauki idan wani saurayi uwa ke shayarwa, a matsayin abu yana da ikon shiga cikin nono madara da kuma isa high yawa a can. Idan alamomi na magani ya kamata a ci gaba, da nono ne mafi alhẽri ga dakatar, ya maye gurbin Na'urar madara cakuda bisa ga yaro ta shekaru.

Side effects da kuma yawan abin sama

Yana iya da illa ga zuciya da jijiyoyin jini, endocrine, urinary, na numfashi, narkewa kamar, kuma tsakiya m tsarin dogon lokacin da amfani da miyagun ƙwayoyi "Sotageksal". Analogs sa irin wannan illa. A haƙuri iya samun:

  • shortness na numfashi, da kara angina harin, cututtuka na zuciya rashin cin nasara, zuciya zafi, vasospasm, Raynaud ta ciwo .
  • tashin zuciya, amai, zawo, ciki zafi, wuce kima gassing, flatulence, da wuya hanji motsi, bushe mucous membranes a bakin.
  • juyayi, agitation, tsoro cuta, hallucinations, illa motor daidaituwa, ji hasara, yanayi swings, tremors, gajiya, ciwon kai, dizziness, rashin barci, ko, conversely, ya karu drowsiness, tashin hankali mafarkai, ciki;
  • conjunctivitis, keratoconjunctivitis, ko bushe ido ciwo (musamman a marasa lafiya da suke ci lambar sadarwa ruwan tabarau kullum), kumburi da cornea, karu a dandano da wari, ido zafi, photophobia, illa gani acuity, ji.
  • da qarancin ruwa da (a mutane da ciwon sukari).
  • bronchospasm, laryngitis, tracheitis.
  • urticaria, dermatitis, fata itching, erythema, psoriasis, angioedema, ta ƙara sweating.
  • namiji iko ciki, ciwo a lokacin kawowa,, mata - rage libido da hailar cuta.
  • zazzabi, tsoka rauni, convulsions, cyanosis na extremities.

A hali na yawan abin sama na iya faruwa:

  • danniya na cardiac ayyuka.
  • shortness na numfashi;
  • asystole, aka rufe da mãgãgi, wani rauni, dizziness.
  • cyanosis na extremities.
  • tsoka cramps.
  • bradycardia zuwa cikakken sakamakon bugun zuciya.
  • zuciya da jijiyoyin jini buga.
  • bronchospasm.
  • tachycardia.

Duk da irin tsanani bayyanar cututtuka na yawan abin sama, mutuwa ne rare. Lokacin da miyagun ƙwayoyi guba farko bukatar dakatar da shan magani "Sotageksal". Analogs da generics sotalol hydrochloride nagarta sosai fitarwa daga gastrointestinal fili bayan ingestion absorbent kwayoyi. A hali na yawan abin sama symptomatic magani aka nuna. A lokuta da tsanani da guba dole ciki lavage da amai, kula da muhimmanci rayuwa da ayyuka na kayan ciki. Wuce kima allurai an cire gaba daya ta hanyar hemodialysis. Rayuwa ragewan jini sugar na iya faruwa a marasa lafiya da suke bi don wani m rage cin abinci ko jin matsananciyar yunwa.

Analogs da generics "Sotageksala"

Sotalol hydrochloride dauke a cikin samfurin samar a Switzerland da Jamus, karkashin cinikin sunan "Sotageksal". Analogues daga gare aka nuna da kuma sauran kwayoyi da daban-daban abun da ke ciki, wanda a Bugu da kari zuwa wani antiarrhythmic sakamako taimaka tsoka spasms, rage hawan jini da kuma inganta aiki na atria. Wadannan sun hada da:

  • "Inderal" "Inderal", "obzidan", "Pranolol" (aiki sashi - propranolol) amfani domin lura da ischemia, arrhythmia da hauhawar jini.
  • "Pumpan" - homeopathic wakili bisa kayan gyara.
  • "Magnerot" ya ƙunshi magnesium orotate dihydrate aka yi amfani ga zalunta arteriosclerosis, cuta na sia metabolism.
  • "Korvitol" (metoprolol tartrate) ne tasiri ga migraines.
  • "Nebilet" (nebivolol hydrochloride) da aka nuna ga hauhawar jini, ischemic cuta.
  • "Qudesan" (drop) - a nazarin halittu kari bisa coenzyme Q10 domin yin rigakafi da magani daga arrhythmias.
  • "Etatsizin" (etatsizin) ne amfani a tachycardia.
  • "Arrhythmia" "Amiodarone" (amiodarone hydrochloride) ana amfani da cardiac, tachycardia, atrial arrhythmia.
  • "Propanorm" (propafenone hydrochloride) da ake amfani da lokacin da na ramin zuciya da kuma supraventricular arrhythmias.
  • "Neo-Giluritmal" (praymaliya bitartrate) da aka nuna ga na ramin zuciya arrhythmias, tachycardia.
  • "Korgard" (nadolol) yana soma domin lura da angina pectoris, migraine.

Rasha samar "Sotalol Canon" da "Tenzol" tare da wannan aiki sashi a matsayin "Sotageksal". Analogues a Moldova, Ukraine da kuma kasashe makwabta a Pharmacy wuta fiye da asali miyagun ƙwayoyi. The kudin da kwayoyi dogara a kan kasar da kuma masu sana'anta. Domestic magunguna yawanci suna da wani farashin muhimmanci ƙananan fiye da waje.

reviews

Akwai wani gagarumin raguwa a kãmun mita a lokacin atrial fibrillation, idan dauka ci gaba "Sotageksal". Analogs haƙuri sake dubawa ba haka ba ne tabbatacce. Shi ne ba ko da yaushe kwayoyi daga daban-daban masana'antun ne irin wannan, har ma idan suna da wannan abun da ke ciki. Mutane da yawa tsõron unscrupulous masana'antun nuna mafi taro na aiki sashi da kwamfutar hannu fiye da akwai zahiri ne. Saboda wannan magani ba zai iya kawo sa ran sakamakon. Reviews na "Sotageksale", da bambanci, mafi kyau. Ya kamata a yi amfani da hadaddun lura da cututtuka na zuciya da cututtuka a matakai daban-daban.

A mafi yawan lokuta akwai karɓa mai kyautata a cikin janar jihar da marasa lafiya batun hadaddun magani. Da miyagun ƙwayoyi ne ba makawa biyu a cupping, da kuma rigakafin. Kuna hukunta da sake dubawa na marasa lafiya tare da ganewar asali "paroxysmal fibrillation," da magani taimaka wajen ci gaba da al'ada zuciya kari (bayar, idan dauka ci gaba kamar yadda tabbatarwa far). Duk da haka, marasa lafiya ce cewa bai yi kuskure tada nasu kashi ba tare da wani likita ta shawarwarin saboda hadarin gaske illa.

Wasu daga cikin sake dubawa ba sosai tabbatacce sakamako a kan suna daga cikin miyagun ƙwayoyi. An yi imani da cewa shi ne tallata da kuma ba zai iya warkar da anemia, da ake dasu arrhythmias, hypokalemia da hypomagnesemia. An lura da cewa sotalol hydrochloride waje brands da wuya a sami a gida Pharmacy. Mutane saba ko da yaushe amfani a wajen fuskantar matsaloli tare da saye. Saboda haka, kafin fara jiyya, tabbatar da cewa shi ba za su iya ci gaba da na dogon lokaci.

Abin da ba za a iya hada liyafar "Sotageksala"

A lokacin jiyya da marasa lafiya shi ne kyawawa su daina tuki, hawan keke, babur. Har ila yau hatsari ne dukkan ayyukan da bukatar ya karu da hankali da kuma psychomotor taro da kuma mayar da hankali. Lokacin da samun ƙarin kudi ga rage matsin lamba ne wata ila don hypotension. An haramta hada "Sotageksal" da irin wannan kwayoyi:

  • insulin, kamar yadda riga qara ta maida hankali a cikin jini.
  • ions da alli antagonists.
  • yana nufin ga general ko inhalation m.
  • Mao hanawa.
  • aidin-dauke da abu.
  • diuretics.
  • ergot alkaloids.
  • tetracyclic antidepressants.

A magani ba anyishi lokaci guda tare da antiarrhythmics na aji na da III. Haka kuma an contraindicated a samun narcotic kwayoyi, sedatives da antihistamines, antipsychotics, coumarin, relaxants. Sun kuma taimaka wa karfi tsakiya m tsarin ciki. Lokaci daya maganin sa barci take kaiwa zuwa ƙãra jini da kuma depresses tsokar nama. An haramta yin wani fata gwajin domin sanin iri allergens. Wannan na kara hadarin anaphylaxis, angioedema, kuma asphyxia.

Drug "Sotageksal" saki a Pharmacy ta sayen magani. Raba magani daga arrhythmia cewa yana iya jawo babbar illa halayen. Saboda haka, kafin ka kai da magani, ya kamata ka ko da yaushe tuntubar likita.

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