Kiwon lafiya, Shirye-shirye
"Theophylline": umarnin don amfani. "Theophylline": alamomi ga yin amfani da analogues
Idan wani mutum ne yake shan wahala daga airway toshewa, wannan mai yiwuwa nuna gaban kullum obstructive na huhu cuta (COPD). Wannan cuta ne quite na kowa. Sau da yawa da ya faru na wannan cuta gani a Club. A ci gaba da wannan cuta ne ya sa ta kamuwa da cuta hit, ko abin da wasu huhu lalacewa. A mutumin da airway constriction iya wuya exhale.
description
"Theophylline", wanda abun da ke ciki za a iya bayyana a kasa, shi ne wani fari crystalline foda. Shi ne dan kadan mai narkewa a cikin ruwan sanyi (a cikin rabo 1: 180), amma an sauƙi narkar da a cikin ruwan zafi (a cikin wani rabo daga 1:85). Yana kuma dissolves a alkalis kuma acid.
tsarin
A wannan halitta da babban aiki sashi ne theophylline. nan kuma sun hada da wasu karin aka gyara. Wato - lactose monohydrate, magnesium stearate, talc, methacrylic acid.
saki Form
Akwai da dama jinsunan a wannan batun. "Theophylline" kerarre a matsayin ci-saki Allunan (0.1 g, 0.25 g), capsules (0.125 g, 0.5 g), da kuma suppositories (0.2 g).
pharmacological ayyuka
Ayyuka na ce halitta ne Multi-faceted. "Theophylline", reviews daga waxanda suke da kyau, shakatawa bada tsokoki na bronchi, yana da wani stimulating da vasodilator mataki. Wannan shiri na tabbatar da al'ada aiki na numfashi cibiyar. Kashe zafi a cikin diaphragm da kuma inganta aiki na intercostal tsokoki kuma taimaka wa "Theophylline". Its amfani a yau da kullum hanya rage yiwuwar bayyanuwar rashin lafiyan halayen a cikin numfashi tsarin irin jikinsu. Ya ce shirye-shiryen da za su iya exert wani diuretic sakamako. A gaban da aiki abubuwa a cikin medicament inganta daidaita numfashi aiki, rage matakin na carbon dioxide, kuma Ya ƙãra iska.
alamomi
Raba-aiki ya ce miyagun ƙwayoyi a faru na Bronchial fuka, asthmatic matsayi, obstructive mashako, na huhu emphysema. Har ila yau, an yi amfani a matsayin agaji a jariri jarirai da apnea. Yi amfani da "Theophylline" da farko a matsayin bronchodilator.
Cikakken bayanin da bakan ce halitta
Da farko, a lura da COPD ne aiki bronchodilators. Sun kawo tonawa Airways. Daya daga cikin wadannan kwayoyi, kamar yadda riga aka ambata a sama, wannan shiri ne a matsayin "theophylline". Umurnai na amfani characterizes shi a matsayin bronchodilator miyagun ƙwayoyi, wanda daukawa fitar da ake kira tarewa na purine rabe. A gaban irin wannan tasiri inji tabbatar da kau da spasms a cikin m tsoka na bronchi, da kawar da zafi a cikin diaphragm, kunnawa da oxygen zuwa huhu, inganta aikin intercostal tsokoki. A sakamakon haka, da Airways bude, mutumin da numfashi sauki.
Yana yana da wani tabbataccen amfani, "Theophylline". Umurnai na amfani na nuni da cewa wannan magani zai iya gaskiya ma tasiri ba kawai a kan numfashi fili, amma kuma a kan sauran jiki tsarin. Wannan magani taimaka wajen fadada jijiyoyin zuciya da kuma na gefe jini, impedes aiwatar da platelet mannewa, shi ne m diuretic mataki. Yana bayar da ruri pruning ayyuka na zuciya tsoka (myocardium), m jini, kazalika da amfani tasiri a kan ta tsakiya m tsarin. A sakamakon haka, da miyagun ƙwayoyi ne iya aiki m, a lokaci guda da ciwon antiasthmatic, bronchodilator, diuretic, spasmolytic, vasodilatory da cardiotonic Properties.
"Theophylline": umarnin don amfani da
Domin sanin da sashi, akwai mutane da yawa sharudda. "Theophylline", bisa ga umarnin, akwai buƙatar ka kai da yara to da shekaru 14 da kuma manya, 300 MG da rana 2-3 sau. A wannan yanayin, da magani ya kamata in sha ruwa a cikin manyan yawa. Idan ya cancanta, da kashi za a iya ƙara zuwa 500 MG sau 2 a rana, idan da shawarar da ka likita. Idan haƙuri yana da jiki nauyi kasa da 60 kg, da sashi ya zama 100 MG sau 2 a rana. A wannan yanayin, da nada sãfe da maraice liyafar da wannan shiri a matsayin "Theophylline". Umarni ya furta cewa, magani wajibi ne a fara da kananan allurai da hankali ƙãra musu zama.
Shan da miyagun ƙwayoyi a lokacin daukar ciki da kuma nono
"Theophylline" sakamako a kan tayin karkashin category "C" ta FDA. A kayan aiki ratsa cikin placental shãmaki. Mata masu ciki da za a iya ce da miyagun ƙwayoyi ne kawai a lokuta inda sa ran amfani zuwa ga uwar shi ne mafi girma daga hadarin m zuwa tayin. A lokacin da na trimester da na karshe makonni na ciki tafii da miyagun ƙwayoyi, lura m alamomi. Yana da muhimmanci a tuna.
Na da yawa lura bayar da shawarar cewa theophylline yarda a lokacin III trimester na ciki da aka rage. Wannan na iya bukatar karin m tabbatar da dalilin da taro na dũkiyõyinsu a jini da kuma wani yiwu rage daga cikin kashi.
Nono "Theophylline" da dama a cikin madara da kuma na iya haifar da cututtuka da irritability a jarirai ko wasu alamu na yawan guba. Yana da muhimmanci a san. A taro na ce abu a nono madara ne kamar daidai da abun ciki a cikin jini magani na uwa. Har ila yau, wannan na nufin muhimmanci damuarn igiyar ciki contractions.
contraindications
"Theophylline" umarnin don amfani da kamar yadda aka bayyana a sama, an contraindicated idan akwai:
- Idiosyncrasy.
- Hyperthyroidism.
- M tsokar zuciya infarction.
- Subaortic stenosis. Wannan shi ne wani ba mai kumburi cuta na hagu ventricle na zuciya tsoka nama. An halin magana da wani kaifi takaita da ta kogo.
- Arrythmia.
- Epilepsy da sauran convulsive yanayi.
- Pregnancy.
Tare da kula da shi wajibi ne don tsayar da liyafar da miyagun ƙwayoyi a lokacin bayyanuwar ulcerative cuta na ciki da kuma duodenum.
takamaiman sharudda
Shan taba muhimmanci rinjayar da gudanar da metabolism da kuma tukar tumbi da irin wannan abubuwa irin theophylline. Ya kamata a tuna. Mutane masu kyafaffen 1-2 fakitoci na taba wata rana, da rage yawan rabin-rai lokaci. A marasa lafiya da hanta, cardiac ko numfashi gazawar bayyana, kazalika da kwayar cututtuka da kuma hyperthermia auku deceleration kawar da aiki abu. Yanayin aiki barasa da kuma maganin kafeyin-type kayayyakin ma yana da wani gagarumin sakamako a kan metabolism na theophylline.
hulda
Da miyagun ƙwayoyi "Theophylline" inganta potentiation sakamako na β2-agonists. Yana kuma iya bunkasa tremor, wanda aka sa ta a sympathomimetic miyagun ƙwayoyi da irin da yake iya hana aiwatar da sha na phenytoin. Slow kawar da nufin ya auku a cikin hulda da "erythromycin" da "phenobarbital." Na nufin "Theophylline" samar da wani karuwa a koda tukar tumbi da lithium. A wannan yanayin, da warkewa balance ne gaji da damuwa a marasa lafiya da suke shan m salts. Da miyagun ƙwayoyi "cimetidine" na taimaka wa taro a cikin jinin theophylline matakan, kuma qara lokacin ta janye. Magunguna da irin wannan illa da za a jera a kasa.
A gaban gefen effects
Lokacin karbar ce kwayoyi iya daban-daban korau bayyanar cututtuka. wato:
- Za ka iya samun bayyanar cututtuka na dizziness, rashin barci, ciwon kai, rufe da mãgãgi, juyayi, tremor, da ruɗewa, epilepsy.
- A cikin zuciya da jijiyoyin jini tsarin - arrhythmia, tachycardia, ƙarya angina, kwatsam karu a jini, angina pectoris.
- Daga cikin narkewa kamar tsarin - fitowan da tashin zuciya da amai, ƙwannafi, zawo, flatulence, colitis, gastritis.
- Lokacin da wajibi na liyafar nufin za a iya lura da wasu bayyananen na rashin lafiyan halayen a cikin nau'i na itching, kona, urticaria, dermatitis, zazzabi, sweating da kuma fata rashes.
yawan abin sama
A wannan yanayin, akwai wasu cututtuka. A karkashin wadannan manifestations unsa:
- agitation.
- rikice.
- convulsions.
- tachycardia.
- arrhythmia.
- hypotension.
- tashin zuciya.
- zawo.
- amai da wani admixture na jini.
- hyperglycemia.
- rayuwa acidosis.
Lokacin da wadannan cututtuka da ake sa wani magani. Wato, za'ayi da:
- Kunna gawayi Hanyar.
- Ban ruwa yankin hanji hade da salts da polyethylene glycol bayani.
- Igiyar jini liyafar "MCP" ko "Ondansetron" da alama bayyanar cututtuka na tashin zuciya da kuma amai.
- Yanayin aiki "benzodiazepines", "Phenobarbital" (ko thiopental sodium) da kuma na gefe tsoka relaxants a faru na seizures.
"Theophylline": takwarorinsu
Akwai da dama daban-daban kwayoyi na irin wannan. A wannan yanayin, ka yi la'akari da wadannan magunguna:
- "Teobiolong" ( "Theobilongum").
- "Spofillinretard" "(Spophillin retard").
- "Perfillon" ( "PerphyUon").
- "Neoefrodal" ( "Neo-Efrodal").
- "Franol" ( "Franol").
ajiya
A powders da Allunan ( "theophylline") adana a wani duhu, bushe wuri. Su shiryayye rayuwa shi ne shekaru biyar. Storage kyandirori ya kamata a yi a cikin firiji. A lokaci guda ya kamata su ba za a daskarewa. Su shiryayye-rai na shekaru hudu.
sakamakon
Bayan karanta a sama, wanda zai iya tunanin abin da wani magani kamar "theophylline", farashin wanda yake m (a cikin 70-160 goga.). Har ila yau a cikin wannan rubutu gaya game da umarnin don amfani da miyagun ƙwayoyi da kuma ta hulda da wasu hanyoyi.
Similar articles
Trending Now